Acid Reflux Medications: Prescription and OTC Proton Pump Inhibitors and H2 Blockers for GERD

Acid reflux — including gastroesophageal reflux disease (GERD), peptic ulcer disease, erosive esophagitis, and related conditions — is among the most common gastrointestinal complaints treated in primary care. Pharmacological management aims to reduce gastric acid secretion, protect the mucosal lining, and allow healing of acid-damaged tissues.

The two primary drug classes are:

  • Proton Pump Inhibitors (PPIs) — the most potent acid-suppression agents, blocking the H+/K+-ATPase pump in gastric parietal cells. Include omeprazole, esomeprazole, lansoprazole, pantoprazole, and rabeprazole. Several are OTC at low doses; all are available at higher doses by prescription.
  • H2 Receptor Antagonists (H2 blockers) — older class; block histamine H2 receptors on parietal cells to reduce acid secretion. Include famotidine (Pepcid) and cimetidine (Tagamet). Note: ranitidine (Zantac) was withdrawn from US and global markets in 2020.

Misoprostol (Cytotec) is a distinct medication also included here — a synthetic prostaglandin used to protect the gastric mucosa when patients must take NSAIDs long-term, and also used for obstetric indications.

Acid Reflux Medications Available at Lucas Clinic

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